Description
α-Helical CRF(9-41) TFA is a competitive CRF2 receptor antagonist with K B of ~100 nM. α-Helical CRF(9-41) TFA is also a partial agonist of CRF1 receptor with an EC 50 of 140 nM.Appearance:SolidIC50& Target:KB: ~100 nM (CRF2 receptor) EC50: 140 nM (CRF1 receptor)Biological Activity:α-Helical CRF(9-41) TFA is a competitive CRF2 receptor antagonist with K B of ~100 nM. α-Helical CRF(9-41) TFA is also a partial agonist of CRF1 receptor with an EC 50 of 140 nM