Description
β-Melanocyte Stimulating Hormone (MSH), human TFA, a 22-residue peptide, acts as an endogenous melanocortin-4 receptor ( MC4-R ) agonist.Appearance:SolidIC50& Target:Melanocortin-4 receptor (MC4-R)In Vitro:β-Melanocyte Stimulating Hormone (MSH), human (β-MSH) has high affinity at both human MC4-R transfected into CHO cells (K i =11.4±0.4 nM) and MC4-R in rat hypothalamic homogenates (K i =5.0±0.4 nM). MCE has not independently confirmed the accuracy ofBiological Activity:β-Melanocyte Stimulating Hormone (MSH), human TFA, a 22-residue peptide, acts as an endogenous melanocortin-4 receptor ( MC4-R ) agonist