Description
(R,R)-CPI-1612 is the isomer of CPI-1612, and can be used as an experimental control. CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC 50 of 8.1 nM for EP300 HAT. CPI-1612 has an anticancer activity